摘要:环氧合酶(Cyclooxygenase,COX)是花生四烯酸(AA)代谢过程中调节前列腺素(prostaglandin,PGs)合成的一种重要的限速酶,也是非类固醇抗炎药(nonsteroidal anti-in-flammatory drugs,NSAID)作用的靶酶。国内外资料已证实其有3种亚型:COX-1、COX-2和COX-3。COX-1被认为是“看家”基因,几乎在所有正常组织中结构性地表达,主要参与维持细胞结构的完整性。
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